RTU Research Outputs and Resources: Reasearch Staff

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors
(2020)

Aiga Grandane, Alessio Nocentini, Thomas Werner, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

7-Acylamino-3H-1,2-benzoxathiepine 2,2-Dioxides as New Isoform-Selective Carbonic Anhydrase IX and XII Inhibitors
(2020)

Aleksandrs Pustenko, Alessio Nocentini, Anastasija Balašova, Mikhail Krasavin, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Sulfocoumarins as Dual Inhibitors of Human Carbonic Anhydrase Isoforms IX/XII and of Human Thioredoxin Reductase
(2020)

Mikhail Krasavin, Raivis Žalubovskis, Aiga Grandane, Ilona Domračeva, Petr Zhmurov, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

The Antibiotic Furagin and Its Derivatives are Isoform-Selective Human Carbonic Anhydrase Inhibitors
(2020)

Aleksandrs Pustenko, Alessio Nocentini, Paola Gratteri, Alessandro Bonardi, Igor Vozny, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Combining Carbonic Anhydrase and Thioredoxin Reductase Inhibitory Motifs within a Single Molecule Dramatically Increases Its Cytotoxicity
(2020)

Mikhail Krasavin, Tatiana Sharonova, Vladimir Sharoyko, Daniil Zhukovsky, Stanislav Kalinin, Raivis Žalubovskis, Tatiana Tennikova, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with Effective Carbonic Anhydrase Inhibitory Activity: Solution and Crystallographic Investigations
(2017)

Jekaterīna Ivanova, Agnese Balode, Raivis Žalubovskis, Janis Leitans, Andris Kazaks, Daniela Vullo, Kaspars Tārs, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

N-Substituted and Ring Opened Saccharin Derivatives Selectively Inhibit Transmembrane, Tumor-Associated Carbonic Anhydrases IX and XII
(2017)

Jekaterīna Ivanova, Fabrizio Carta, Daniela Vullo, Janis Leitans, Andris Kazaks, Kaspars Tārs, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

CCDC 1526002: Experimental Crystal Structure Determination
(2017)

Aleksandrs Pustenko, Dmitrijs Stepanovs, Raivis Žalubovskis, Daniela Vullo, Andris Kazaks, Janis Leitans, Kaspars Tārs, Claudiu T. Supuran
Internet publication

X-Ray Crystallography-Promoted Drug Design of Carbonic Anhydrase Inhibitors
(2015)

Jekaterīna Ivanova, Raivis Žalubovskis, Muhammet Tanc, Andris Kazaks, Claudiu T. Supuran, Kaspars Tārs, Janis Leitans
Scientific article indexed in SCOPUS or WOS database

Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX
(2015)

Jekaterīna Ivanova, Agnese Balode, Raivis Žalubovskis, Kaspars Tārs, Andris Kazaks, Janis Leitans, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Information about Author

Publications

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors
(2020)

7-Acylamino-3H-1,2-benzoxathiepine 2,2-Dioxides as New Isoform-Selective Carbonic Anhydrase IX and XII Inhibitors
(2020)

Sulfocoumarins as Dual Inhibitors of Human Carbonic Anhydrase Isoforms IX/XII and of Human Thioredoxin Reductase
(2020)

The Antibiotic Furagin and Its Derivatives are Isoform-Selective Human Carbonic Anhydrase Inhibitors
(2020)

Combining Carbonic Anhydrase and Thioredoxin Reductase Inhibitory Motifs within a Single Molecule Dramatically Increases Its Cytotoxicity
(2020)

5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with Effective Carbonic Anhydrase Inhibitory Activity: Solution and Crystallographic Investigations
(2017)

N-Substituted and Ring Opened Saccharin Derivatives Selectively Inhibit Transmembrane, Tumor-Associated Carbonic Anhydrases IX and XII
(2017)

CCDC 1526002: Experimental Crystal Structure Determination
(2017)

X-Ray Crystallography-Promoted Drug Design of Carbonic Anhydrase Inhibitors
(2015)

Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX
(2015)

Information about Author

Publications

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors (2020)

7-Acylamino-3H-1,2-benzoxathiepine 2,2-Dioxides as New Isoform-Selective Carbonic Anhydrase IX and XII Inhibitors (2020)

Sulfocoumarins as Dual Inhibitors of Human Carbonic Anhydrase Isoforms IX/XII and of Human Thioredoxin Reductase (2020)

The Antibiotic Furagin and Its Derivatives are Isoform-Selective Human Carbonic Anhydrase Inhibitors (2020)

Combining Carbonic Anhydrase and Thioredoxin Reductase Inhibitory Motifs within a Single Molecule Dramatically Increases Its Cytotoxicity (2020)

5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with Effective Carbonic Anhydrase Inhibitory Activity: Solution and Crystallographic Investigations (2017)

N-Substituted and Ring Opened Saccharin Derivatives Selectively Inhibit Transmembrane, Tumor-Associated Carbonic Anhydrases IX and XII (2017)

CCDC 1526002: Experimental Crystal Structure Determination (2017)

X-Ray Crystallography-Promoted Drug Design of Carbonic Anhydrase Inhibitors (2015)

Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX (2015)

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors
(2020)

7-Acylamino-3H-1,2-benzoxathiepine 2,2-Dioxides as New Isoform-Selective Carbonic Anhydrase IX and XII Inhibitors
(2020)

Sulfocoumarins as Dual Inhibitors of Human Carbonic Anhydrase Isoforms IX/XII and of Human Thioredoxin Reductase
(2020)

The Antibiotic Furagin and Its Derivatives are Isoform-Selective Human Carbonic Anhydrase Inhibitors
(2020)

Combining Carbonic Anhydrase and Thioredoxin Reductase Inhibitory Motifs within a Single Molecule Dramatically Increases Its Cytotoxicity
(2020)

5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with Effective Carbonic Anhydrase Inhibitory Activity: Solution and Crystallographic Investigations
(2017)

N-Substituted and Ring Opened Saccharin Derivatives Selectively Inhibit Transmembrane, Tumor-Associated Carbonic Anhydrases IX and XII
(2017)

CCDC 1526002: Experimental Crystal Structure Determination
(2017)

X-Ray Crystallography-Promoted Drug Design of Carbonic Anhydrase Inhibitors
(2015)

Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX
(2015)