RTU Research Outputs and Resources: Reasearch Staff

Thiochromenocarbazole Imide-Based Photosensitizers Decorated with Carbonic Anhydrase Inhibitors for the Targeted Treatment of Hypoxic Tumours
(2024)

Amina Merabti, Dario Puchan Sanchez, Alessio Nocentini, Lamiaa M A Ali, Christophe Nguyen, Denis Durand, Kathleen Haman, Tatiana Ghanem, Phillippe Arnoux, Pierre Josse, Celine Frohot, Raivis Žalubovskis
Scientific article indexed in SCOPUS or WOS database

1,2,3-Benzoxathiazine-2,2-Dioxides–Effective Inhibitors of Human Carbonic Anhydrases
(2023)

Jekaterīna Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

3H-1,2-Benzoxaphosphepine 2-Oxides as Selective Inhibitors of Carbonic Anhydrase IX and XII
(2023)

Aleksandrs Pustenko, Anastasija Balašova, Alessio Nocentini, Claudiu T. Supuran, Raivis Žalubovskis
Scientific article indexed in SCOPUS or WOS database

Derivatives of 4-Methyl-1,2,3-benzoxathiazine 2,2-Dioxide as Selective Inhibitors of Human Carbonic Anhydrases IX and XII over the Cytosolic Isoforms I and II
(2023)

Jekaterīna Ivanova, Morteza Abdoli, Alessio Nocentini, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect
(2023)

Jekaterīna Ivanova, Alessio Nocentini, Kaspars Tārs, Janis Leitans, Elviss Dvinskis, Andris Kazaks, Ilova Domračeva, Claudiu T. Supuran, Raivis Žalubovskis
Scientific article indexed in SCOPUS or WOS database

Aryl Derivatives of 3H-1,2-Benzoxaphosphepine 2-Oxides as Inhibitors of Cancer-Related Carbonic Anhydrase Isoforms IX and XII
(2023)

Anastasija Balašova, Aleksandrs Pustenko, Alessio Nocentini, Daniela Vullo, Claudiu T. Supuran, Raivis Žalubovskis
Scientific article indexed in SCOPUS or WOS database

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors
(2021)

Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Žalubovskis, valentina Onnis, Wagdy E. Eldehna, Clemente Capasso, Simone Carradori, William A. Donald, Shoukat Dedhar, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment
(2020)

Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Žalubovskis, Atilla Akdemir, valentina Onnis, Wagdy E. Eldehna, Clemente Capasso, Giuseppina De Simone, Simona Maria Monti, Simone Carradori, William A. Donald, Shoukat Dedhar, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Development of Oxathiino[6,5-b]pyridine 2,2-Dioxide Derivatives as Selective Inhibitors of Tumor-Related Carbonic Anhydrases IX and XII
(2020)

Aiga Grandane, Alessio Nocentini, Ilona Domračeva, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors
(2020)

Aiga Grandane, Alessio Nocentini, Thomas Werner, Raivis Žalubovskis, Claudiu T. Supuran
Scientific article indexed in SCOPUS or WOS database

Information about Author

Publications

Thiochromenocarbazole Imide-Based Photosensitizers Decorated with Carbonic Anhydrase Inhibitors for the Targeted Treatment of Hypoxic Tumours
(2024)

1,2,3-Benzoxathiazine-2,2-Dioxides–Effective Inhibitors of Human Carbonic Anhydrases
(2023)

3H-1,2-Benzoxaphosphepine 2-Oxides as Selective Inhibitors of Carbonic Anhydrase IX and XII
(2023)

Derivatives of 4-Methyl-1,2,3-benzoxathiazine 2,2-Dioxide as Selective Inhibitors of Human Carbonic Anhydrases IX and XII over the Cytosolic Isoforms I and II
(2023)

Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect
(2023)

Aryl Derivatives of 3H-1,2-Benzoxaphosphepine 2-Oxides as Inhibitors of Cancer-Related Carbonic Anhydrase Isoforms IX and XII
(2023)

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors
(2021)

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment
(2020)

Development of Oxathiino[6,5-b]pyridine 2,2-Dioxide Derivatives as Selective Inhibitors of Tumor-Related Carbonic Anhydrases IX and XII
(2020)

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors
(2020)

Patents

4-((5-substituted-4-OXO-4,5-dihydrothiazol-2-YL)amino)benzenesulfonamide derivatives as potential agents for neuropathic pain
LV15831B (20.04.2025.)

Information about Author

Publications

Thiochromenocarbazole Imide-Based Photosensitizers Decorated with Carbonic Anhydrase Inhibitors for the Targeted Treatment of Hypoxic Tumours (2024)

1,2,3-Benzoxathiazine-2,2-Dioxides–Effective Inhibitors of Human Carbonic Anhydrases (2023)

3H-1,2-Benzoxaphosphepine 2-Oxides as Selective Inhibitors of Carbonic Anhydrase IX and XII (2023)

Derivatives of 4-Methyl-1,2,3-benzoxathiazine 2,2-Dioxide as Selective Inhibitors of Human Carbonic Anhydrases IX and XII over the Cytosolic Isoforms I and II (2023)

Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect (2023)

Aryl Derivatives of 3H-1,2-Benzoxaphosphepine 2-Oxides as Inhibitors of Cancer-Related Carbonic Anhydrase Isoforms IX and XII (2023)

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors (2021)

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment (2020)

Development of Oxathiino[6,5-b]pyridine 2,2-Dioxide Derivatives as Selective Inhibitors of Tumor-Related Carbonic Anhydrases IX and XII (2020)

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors (2020)

Patents

4-((5-substituted-4-OXO-4,5-dihydrothiazol-2-YL)amino)benzenesulfonamide derivatives as potential agents for neuropathic pain LV15831B (20.04.2025.)

Thiochromenocarbazole Imide-Based Photosensitizers Decorated with Carbonic Anhydrase Inhibitors for the Targeted Treatment of Hypoxic Tumours
(2024)

1,2,3-Benzoxathiazine-2,2-Dioxides–Effective Inhibitors of Human Carbonic Anhydrases
(2023)

3H-1,2-Benzoxaphosphepine 2-Oxides as Selective Inhibitors of Carbonic Anhydrase IX and XII
(2023)

Derivatives of 4-Methyl-1,2,3-benzoxathiazine 2,2-Dioxide as Selective Inhibitors of Human Carbonic Anhydrases IX and XII over the Cytosolic Isoforms I and II
(2023)

Atropo/Tropo Flexibility: A Tool for Design and Synthesis of Self-Adaptable Inhibitors of Carbonic Anhydrases and Their Antiproliferative Effect
(2023)

Aryl Derivatives of 3H-1,2-Benzoxaphosphepine 2-Oxides as Inhibitors of Cancer-Related Carbonic Anhydrase Isoforms IX and XII
(2023)

Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors
(2021)

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment
(2020)

Development of Oxathiino[6,5-b]pyridine 2,2-Dioxide Derivatives as Selective Inhibitors of Tumor-Related Carbonic Anhydrases IX and XII
(2020)

Benzoxepinones: A New Isoform-Selective Class of Tumor Associated Carbonic Anhydrase Inhibitors
(2020)

4-((5-substituted-4-OXO-4,5-dihydrothiazol-2-YL)amino)benzenesulfonamide derivatives as potential agents for neuropathic pain
LV15831B (20.04.2025.)